Nab-rapamycin (** Currently investigational - no approved brand names available. Developed by Aadi Biosciences under the designation ABI-009. **)

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Description

Nab-rapamycin (also known as ABI-009) is an investigational drug currently being studied in clinical trials. It is a type of mTOR inhibitor. In the context of colorectal cancer, it has been studied in combination with nivolumab (Opdivo) in patients with advanced MSI-H/dMMR metastatic colorectal cancer. The goal of the clinical trial (NCT03190174) was to determine the maximum safe dose of nab-rapamycin when given after nivolumab and to see how effective this combination is in controlling the cancer and extending the time without disease progression (progression-free survival). It is important to note that this drug is still in early-phase trials and is not yet approved for treating colorectal cancer or any other cancer.

Mechanism of Action

Nab-rapamycin is an mTOR inhibitor. mTOR (mammalian target of rapamycin) is a protein that plays a key role in cell growth, division, and survival. By inhibiting mTOR, nab-rapamycin aims to block these processes in cancer cells, potentially slowing or stopping their growth. In the trial mentioned, it was used in combination with nivolumab, an immunotherapy drug that helps the immune system recognize and attack cancer cells. The combination aims to target both the cancer cells directly (via mTOR inhibition) and stimulate the immune system against them.

Side Effects

As nab-rapamycin is an investigational drug in early-phase trials The full range of potential side effects is still being evaluated. Clinical trials are designed to carefully monitor patients for side effects and determine the drug's safety profile. Common side effects associated with mTOR inhibitors can include fatigue Rash Diarrhea Mouth sores And changes in blood counts. Specific side effects observed in the NCT03190174 trial involving nab-rapamycin and nivolumab are being assessed But detailed information is not yet widely available. Patients participating in clinical trials are closely monitored for any adverse events.

Not all side effects are listed. Side effects vary by individual. Always consult your oncologist.

Clinical Trials

NCT03190174 med_phase_prefix1
Archived
Nivolumab (Opdivo®) Plus ABI-009 (Nab-rapamycin) for Advanced Sarcoma and Certain Cancers
United States