Darlifarnib

Targeted Therapy

Description

Darlifarnib is under investigation for its potential role in the treatment of colorectal cancer; it has shown promise in preclinical models and early-phase clinical trials as a targeted therapy against tumors with aberrant Hedgehog pathway activation; however, further research is needed to establish its efficacy and safety profile specifically in colorectal cancer patients.

Mechanism of Action

Darlifarnib is a selective inhibitor of the SMO protein, which plays a critical role in the Hedgehog signaling pathway; this pathway is often aberrantly activated in various cancers including colorectal cancer, contributing to tumor growth and survival.

Side Effects

Fatigue; nausea; diarrhea; increased blood pressure; headache

Not all side effects are listed. Side effects vary by individual. Always consult your oncologist.

Clinical Trials

NCT06026410 Phase 1
Recruiting
KO-2806 Monotherapy and Combination Therapies in Advanced Solid Tumors
United States, France, Germany, Italy, Spain